Drug interactions with Methylphenidate

Drug class
Drugs
Interaction
Adrenergic neurone blockers
Debrisoquine, guanethidine, bretylium.
Antagonism of hypotensive effects
Antipsychotics
Clozapine, loxapine, olanzapine, oxypertine, risperidone, pimozide
sulpiride, phenothiazines (chlorpromazine, levomepromazine, (methotrimeprazine), promazine, pericyazine
pipotiazine, thioridazine
fluphenazine, perphenazine, prochlorperazine, trifluoperazine), butyrophenones (benperidol, haloperidol) thioxanthenes (flupentixol, zuclopenthixol), amisulpride, quetiapine, zotepine.
Antagonism of pressor action
Clonidine
Clonidine
Serious adverse effects have been reported with concomitant use of methylphenidate and clonidine (e.g. ****), although a causal relationship has not been established and the safety of using a combination of methylphenidate and clonidine has not been evaluated systematically.
Doxapram
Doxapram
Risk of hypertension
MAOIs
Isocarboxazid, Phenelzine, Tranylcypromine.
Risk of hypertensive crisis
(Should not use concomitantly or within 14 days of discontinuation)
Moclobemide
Moclobemide
Risk of hypertensive crisis
Oxytocin
Oxytocin
Hypertension due to enhanced vasopressor effect of vasoconstrictor sympathomimetics
Phenobarbital
Phenobarbital
Possibly increased plasma-phenobarbital and methylphenidate concentration
Phenytoin
Phenytoin
Increased plasma-phenytoin and methylphenidate concentration
Primidone
Primidone
Possibly increased plasma-primidone and methylphenidate concentration
Selective serotonin reuptake inhibitors
Citalopram, fluoxetine, fluvoxamine maleate, paroxetine, sertraline.
Metabolism of SSRI may be inhibited
Tricyclic antidepressants
Amitriptyline, amoxapine, clomipramine, dosulepin (dothiepin), doxepin, imipramine, lofepramine, nortriptyline, trimipramine.
Metabolism of tricyclic may be inhibited
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© 2006 Royal College of Psychiatrists